SYNTHESIS OF BIOLOGICALLY ACTIVE COMPOUNDS AND STUDY OF THEIR PHARMACOLOGICAL ACTIVITY
Abstract
This article examines the synthesis of biologically active compounds and the comprehensive study of their pharmacological activity as a fundamental direction in modern medicinal chemistry. The paper highlights contemporary synthetic strategies used for constructing structurally diverse and functionally optimized molecules, including classical organic synthesis, stereoselective methods, green chemistry approaches, and combinatorial techniques. Special attention is given to the role of structure–activity relationship (SAR) analysis in guiding molecular modification and enhancing therapeutic efficacy.
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